Top Grade Tianeptine Sodium Salt CAS 30123-17-2 for Anti Depression

• CAS No.: 30123-17-2
• Formula: C21h24cln2nao4s
• EINECS: 250-059-3
• Type: Pharmaceutical Intermediates
• Appearance: Powder
• Quality: Refined
• Model NO.: PY202211032108
• Colour: White
• Transport Package: 1kg/Aluminum Bag or 25kg/Drum
• Specification: 99% min
• Trademark: Puya
• Origin: China
• Production Capacity: 5000kilogram/Month

Product Description

Top Grade Tianeptine Sodium Salt CAS 30123-17-2 For Anti Depression

Product Name:    Tianeptine sodium salt
Synonyms:    TIANEPTINE SODIUM;TIANEPTINE SODIUM SALT;7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Ac id S,S-Dioxide Sodium Salt;S-1574;Stablon;7-[(3-chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepine-11-yl)amino]heptanoic ac id s,s dioxide sodium salt;[7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepine 5,5-dioxide)-11-ylamino]heptanoic ac id]sodium salt;3-Chloro-6,11-dihydro-6-methyl-11-[6-(sodiooxycarbonyl)hexylamino]dibenzo[c,f][1,2]thiazepine 5,5-dioxide
CAS:    30123-17-2
MF:    C21H24ClN2NaO4S
MW:    458.93
EINECS:    250-059-3
Product Categories:    chemical;Stablon, Coaxil, Tatinol;Intermediates & Fine Chemicals;Pharmaceuticals;API;Inhibitors;Heterocycles;Sulfur & Seleni um Compounds;Tianeptine sodi;30123-17-2
Mol File:    30123-17-2.mol

Tianeptine sodium salt is a salt of Tianeptine. Tianeptine is an atypical antidepressant. It is an agonist of the μ-opioid receptor (MOR; EC50s = 194 and 641 nM for human and mouse receptors, respectively, in a BRET assay for G protein activation) and also has effects on the glutamate system. Tianeptine (30 mg/kg) decreases immobility in the forced swim test in wild-type, but not MOR knockout mice, indicating antidepressant-like activity dependent on MORs. It increases locomotor activity at a dose of 30, but not 10 mg/kg, in the open field test and increases paw withdrawal latency in the hot-plate test in mice. Tianeptine modulates AMPA receptor activity by increasing phosphorylation of the AMPA receptor GluR1 subunit in the frontal cortex and hippocampal CA3 region in mice. It prevents increases in glial glutamate transporter 1 (GLT-1) expression induced by chronic restraint stress in the hippocampal CA3 region in rats when administered at a dose of 10 mg/kg per day for 21 days.5It also reverses increases in extracellular glutamate levels induced by acute restraint stress in the basolateral nucleus of the amygdala in rats.

Tianeptine Sodium Salt CAS 30123-17-2 of Chemical Properties
Melting point     1800C
storage temp.     Desiccate at RT
solubility     DMSO: ≥20mg/mL
form     solid
color     white to tan
Merck     14,9420
Stability:    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 2 months.
InChIKey    ZLBSUOGMZDXYKE-UHFFFAOYSA-M
SMILES    C1(NCCCCCCC([O-])=O)C2C=CC=CC=2N(C)S(=O)(=O)C2C=C(Cl)C=CC1=2.[Na+]
CAS DataBase Reference    30123-17-2(CAS DataBase Reference)

Function and Application of Tianeptine Sodium Salt CAS 30123-17-2
Tianeptine Sodium Salt, with CAS number 30123-17-2, is a salt form of tianeptine, a pharmaceutical compound that has been used primarily as an antidepressant and anxiolytic agent. Here are some of its functions and applications:

1. Antidepressant: Tianeptine Sodium Salt is mainly used as an antidepressant drug. It works by regulating the levels of certain neurotransmitters in the brain, including serotonin, norepinephrine, and dopamine. By doing so, it can help improve mood, reduce anxiety, and relieve depression symptoms.

2. Anxiolytic: Tianeptine Sodium Salt also has anxiolytic properties, meaning it can help reduce anxiety and stress. It has been found to be particularly effective in treating anxiety disorders such as generalized anxiety disorder (GAD), social anxiety disorder, and post-traumatic stress disorder (PTSD).

3. Neuroprotective: Tianeptine Sodium Salt has been found to have neuroprotective effects, meaning it can help protect brain cells from damage caused by stress, inflammation, and other factors. This may be due in part to its ability to regulate glutamate transmission in the brain.

4. Pain relief: Tianeptine Sodium Salt has been found to have analgesic properties, meaning it can help reduce pain. It may be particularly effective in treating chronic pain conditions such as fibromyalgia and neuropathic pain.

5. Cognitive enhancement: Tianeptine Sodium Salt has been found to have cognitive enhancing properties, meaning it can help improve cognitive function, including memory, attention, and learning. This may be due in part to its effects on glutamate transmission in the brain.


Packing And Shipping
1.Preferentially DHL, FedEX or TNT for quantity less than 50kg, air shipping for 100kg above, sea shipping for quantity over 500kg.
2.For customers from Russia,Mexico,Turkey,Solvenia,Romania,etc,before placing an order,please kindly confirm if you can make clearance when goods reach your customs.

Shipping Terms
By Express	By Air	By Sea
Suitable for under 50kg Fast:3-4 days High cost Door to door service Easy to pick up the goods	Suitable for more than 50kg Fast:3-4 days High cost Airport to airport Professional broker needed	Suitable for more than 500kg Slow:15-30 days Low cost Port to port Professional broker needed

 

Company Profile
Anhui puya biological technology co.,ltd was established in Hefei. Registered capital is 5 million. It is specialized in manufacture plant extract, API and chemicals raw material powder, food additives and oil. which are applied to skin care, healthcare, weight loss products, sex improvement, and pharmaceuticals. We will uphold honesty and pragmatic, innovative and enterprising service purposes, and provide a variety of quality services to our customers at abroad. It aims at supplying good product and comfort service. The strict quality control is to meet the customer's requirement, to get a highly praised and to be high quality supplier. If you have any question, or need samples, please feel free to contact us.

FAQ
Q1. What's the MOQ?
A: Usually 1 kg.  It is based on the different product. Some are 1g and some are 1 ton. Please be free to consult our salesman.
 
Q2. What's the shipping time?
A: If in stock, we will ship it out immediately.  By FedEx will be 3~5 days to you.
 
Q3. If I need less than the MOQ, is it possible?
A: Yes. Please be free to consult our salesman.
 
Q4. Can you supply the free sample?
A: Usually it is possible. but the shipping cost be paid by customers. It based on the different product. Please be free to consult our salesman.
 
Q5. How to store the product?
A: Store in cool and dry place. It must be in well closed containers. The shelf life will be 2 years.
 
Q6: What's your main payment method?
A: T/T, trade assurance, west union, money gram.
 
Q7: Do you have COA, MSDS, CO, Health certificate, form 9 or other certificate?
A: Yes, we have. pls be free to contact us to get updated one.